CID 16020046

CAS No. 834903-43-4

CID 16020046 ( CID16020046; CID-16020046 )

Catalog No. M19158 CAS No. 834903-43-4

CID16020046 is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast.

Purity : 98%

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 50 In Stock
5MG 83 In Stock
10MG 131 In Stock
25MG 221 In Stock
50MG 327 In Stock
100MG 485 In Stock
200MG Get Quote In Stock
500MG Get Quote In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    CID 16020046
  • Note
    Research use only, not for human use.
  • Brief Description
    CID16020046 is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast.
  • Description
    CID16020046 is a selective GPR55 inverse agonist. CID16020046 is a G protein-coupled receptor that is weakly activated by some cannabinoids at nM concentrations. CID16020046 has been shown to block GPR55-mediated endothelial wound healing and reverse LPI-inhibited platelet aggregation.
  • Synonyms
    CID16020046; CID-16020046
  • Pathway
    Others
  • Target
    Other Targets
  • Recptor
    GPR55
  • Research Area
    Others-Field
  • Indication
    ——

Chemical Information

  • CAS Number
    834903-43-4
  • Formula Weight
    425.44
  • Molecular Formula
    C25H19N3O4
  • Purity
    98%
  • Solubility
    DMSO : ≥ 28 mg/mL; 65.81 mM
  • SMILES
    CC1=CC=C(C=C1)C2=NNC3=C2C(N(C3=O)C4=CC=C(C=C4)C(=O)O)C5=CC(=CC=C5)O
  • Chemical Name
    4-[4-(3-hydroxyphenyl)-3-(4-methylphenyl)-6-oxo-1,4-dihydropyrrolo[3,4-d]pyrazol-5-yl]benzoic acid

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Kargl J, et al. A selective antagonist reveals a potential role of G protein-coupled receptor 55 in platelet and endothelial cell function. J Pharmacol Exp Ther. 2013 Jul;346(1):54-66.
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