CID 16020046
CAS No. 834903-43-4
CID 16020046 ( CID16020046; CID-16020046 )
Catalog No. M19158 CAS No. 834903-43-4
CID16020046 is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast.
Purity : 98%
COA
Datasheet
HNMR
HPLC
MSDS
Handing Instructions
Size | Price / USD | Stock | Quantity |
2MG | 50 | In Stock |
|
5MG | 83 | In Stock |
|
10MG | 131 | In Stock |
|
25MG | 221 | In Stock |
|
50MG | 327 | In Stock |
|
100MG | 485 | In Stock |
|
200MG | Get Quote | In Stock |
|
500MG | Get Quote | In Stock |
|
1G | Get Quote | In Stock |
|
Biological Information
-
Product NameCID 16020046
-
NoteResearch use only, not for human use.
-
Brief DescriptionCID16020046 is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast.
-
DescriptionCID16020046 is a selective GPR55 inverse agonist. CID16020046 is a G protein-coupled receptor that is weakly activated by some cannabinoids at nM concentrations. CID16020046 has been shown to block GPR55-mediated endothelial wound healing and reverse LPI-inhibited platelet aggregation.
-
SynonymsCID16020046; CID-16020046
-
PathwayOthers
-
TargetOther Targets
-
RecptorGPR55
-
Research AreaOthers-Field
-
Indication——
Chemical Information
-
CAS Number834903-43-4
-
Formula Weight425.44
-
Molecular FormulaC25H19N3O4
-
Purity98%
-
SolubilityDMSO : ≥ 28 mg/mL; 65.81 mM
-
SMILESCC1=CC=C(C=C1)C2=NNC3=C2C(N(C3=O)C4=CC=C(C=C4)C(=O)O)C5=CC(=CC=C5)O
-
Chemical Name4-[4-(3-hydroxyphenyl)-3-(4-methylphenyl)-6-oxo-1,4-dihydropyrrolo[3,4-d]pyrazol-5-yl]benzoic acid
Shipping & Storage Information
-
Storage(-20℃)
-
ShippingWith Ice Pack
-
Stability≥ 2 years
Reference
1. Kargl J, et al. A selective antagonist reveals a potential role of G protein-coupled receptor 55 in platelet and endothelial cell function. J Pharmacol Exp Ther. 2013 Jul;346(1):54-66.
molnova catalog
related products
-
Moluccanin
Moluccanin is a natural product isolated from Aleurites moluccana.
-
Regaloside D
Regaloside D is a natural product isolated from Lilium Longiflorum.
-
N1,N5,N10-(E)-tri-p-...
N1,N5,N10-(E)-tri-p-coumaroylspermidine shows free radical-scavenging activity.